Stéphane De Cesco

Abstract 4498: Discovery of novel SMARCA2 small molecule inhibitors with best-in-class potency and selectivity for the treatment of SMARCA4-mutant cancers.

Lijs Beke, Sandrine Grosse, Shaun Martin, Godelieve Lammens et autres

be (code pays fourni par la source)

Abstract 4578: Discovery of a Best-in-Class small molecule p53 Y220C reactivator: Breaking through the potency ceiling

Ruben Boon, Jo Alen, Nihed Draoui, Koen Vandyck et autres

be, us (code pays fourni par la source)

A Computational Community Blind Challenge on Pan-Coronavirus Drug Discovery Data

Hugo MacDermott-Opeskin, Jenke Scheen, Cas Wognum, Joshua T. Horton et autres

us, gb, il, cl, ca, lu, cn, cz, de, fr, at, ir, jp, in (code pays fourni par la source)

Abstract C113: Discovery of Best-in-Class FGFR3 small molecule inhibitors with high isoform selectivity and activity against gatekeeper mutations

Sandrine Vendeville, Lijs Beke, Ellen A. Lanckacker, Caroline Joannesse et autres

be (code pays fourni par la source)

Abstract C011: Discovery of novel SMARCA2 small molecule inhibitors with best-in-class potency and selectivity for the treatment of SMARCA4-mutant cancers

Lijs Beke, Sandrine Grosse, Shaun Martin, Godelieve Lammens et autres

be (code pays fourni par la source)

Abstract C012: Discovery of a Best-in-Class small molecule p53 Y220C reactivator: Breaking through the potency ceiling

Ruben Boon, Jo Alen, Nihed Draoui, Koen Vandyck et autres

be (code pays fourni par la source)

A Computational Community Blind Challenge on Pan-Coronavirus Drug Discovery Data

Hugo MacDermott-Opeskin, Jenke Scheen, Cas Wognum, Joshua T. Horton et autres

us, gb, il, cl, ca, lu, cn, cz, de, fr, at, ir, jp, in (code pays fourni par la source)

Design, synthesis and biological evaluation of novel [5,5]-fused thiazolidine/oxazolidine inhibitors for targeting prolyl oligopeptidase

Thershan Satkunarajah, Stéphane De Cesco, Ho Ying Huang, Emmanuelle Nguyen et autres

ca (code pays fourni par la source)

A Computational Community Blind Challenge on Pan-Coronavirus Drug Discovery Data

Hugo MacDermott-Opeskin, Jenke Scheen, Cas Wognum, Joshua T. Horton et autres

us, gb, il, cl, ca, lu, cn, cz, de, fr, at, ir, jp, in (code pays fourni par la source)

A Computational Community Blind Challenge on Pan-Coronavirus Drug Discovery Data

Hugo MacDermott-Opeskin, Jenke Scheen, Cas Wognum, Joshua T. Horton et autres

us, gb, il, cl, ca, lu, cn, cz, de, fr, at, ir, jp, in (code pays fourni par la source)

ChemProp multi-task models for predicting ADME properties in the Polaris challenge

Kenneth Goossens, Giovanni Tricarico, Johan Hofmans, Marie-Pierre Dréanic et autres

Structure elucidation of a human melanocortin-4 receptor specific orthosteric nanobody agonist

Thomas D. Fontaine, Andreas Büsch, Toon Laeremans, Stéphane De Cesco et autres

be, nl, us (code pays fourni par la source)