Accès ouvert
2026
supplementary-materials
OpenAlex
Han Wang, Yuxuan Luo, Sandeep Artham, Qianqian Wang et autres
Supplementary Fig. 6: Comparative pathway analysis reveals distinct transcriptional effects of MTO and fulvestrant
Accès ouvert
2026
supplementary-materials
OpenAlex
Han Wang, Yuxuan Luo, Sandeep Artham, Qianqian Wang et autres
Supplementary Fig. 1: MTO, unlike fulvestrant, maintains E2-mediated ER-SRC3 interaction
Accès ouvert
2026
other
OpenAlex
Han Wang, Yuxuan Luo, Sandeep Artham, Qianqian Wang et autres
Abstract The estrogen receptor (ER or ERα) remains the primary therapeutic target for luminal breast cancer, with current treatments centered on competitive antagonists, receptor downregulators, and aromatase inhibitors. Despite these options, resistance frequently emerges, highlighting the need for alternative targeting strategies. We …
Accès ouvert
2026
supplementary-materials
OpenAlex
Han Wang, Yuxuan Luo, Sandeep Artham, Qianqian Wang et autres
Supplementary Fig. 5: ER protein levels in wild-type and Y537S ER orthotopic xenograft tumors
Accès ouvert
2026
supplementary-materials
OpenAlex
Han Wang, Yuxuan Luo, Sandeep Artham, Qianqian Wang et autres
Supplementary Fig. 2: MTO demonstrates enhanced growth inhibition in endocrine-resistant T47D cells
Accès ouvert
2026
supplementary-materials
OpenAlex
Han Wang, Yuxuan Luo, Sandeep Artham, Qianqian Wang et autres
Supplementary Fig. 7: Comparative transcriptional pathway analysis of MTO and fulvestrant treatments
Accès ouvert
2026
supplementary-materials
OpenAlex
Han Wang, Yuxuan Luo, Sandeep Artham, Qianqian Wang et autres
Supplementary Fig. 3: Three-dimensional spheroid growth in MCF7 cells expressing wildtype and mutant ER
Accès ouvert
2026
supplementary-materials
OpenAlex
Han Wang, Yuxuan Luo, Sandeep Artham, Qianqian Wang et autres
Supplementary Table 1: Analysis of top computational docking candidates from the NIH Clinical Collection
Accès ouvert
2026
supplementary-materials
OpenAlex
Han Wang, Yuxuan Luo, Sandeep Artham, Qianqian Wang et autres
Supplementary Fig. 4: Evaluation of combination treatment effects between MTO and established ER antagonists in MCF7 cells
Accès ouvert
2026
erratum
OpenAlex
Ali Mirtaghavi, Andy Baldwin, Nader Tanideh, Moein Zarei et autres
gb, ir, pl, cn
(code pays fourni par la source)